I-High Purity Pharmaceutical Grade 1421373-66-1 Mesylate-AZD9291 yokwelashwa komdlavuza
Umkhiqizoigama | I-AZD-9291 mesylate |
Omqondofana | N--[2-[[2-(Dimethylamino)ethyl]methylamino]-4-methoxy-5-[[4-(1-methyl-1H-indol-3-yl)-2-pyrimidinyl]amino]phenyl]- 2-propenamide methanesulfonate (1:1) |
Inombolo ye-CAS. | 1421373-66-1 |
Ukubukeka | Impushana eqinile emhlophe ukuya kokuphuzi ngokukhanyayo |
I-Molecular Formula | C28H33N7O2.CH4O3S |
Isisindo samangqamuzana | 595.71 |
Ukusetshenziswa | Ibanga Lezemithi noma inhloso yocwaningo |
Ukupakisha | Njengesicelo sakho |
Isitoreji | Londoloza ezitsheni eziqinile, ezimelana nokukhanya endaweni epholile |
I-AZD-9291 mesylateI-CAS:1421373-66-1 | ||
Items | Sizindinganiso | Rimiphumela |
Ukubukeka | Impushana eqinile emhlophe ukuya kokuphuzi ngokukhanyayo | Impushana eqinile ephuzi ngokukhanyayo |
Iukuhlonza | Ibhalwe ngu-IR | Iyahambisana |
Nge-HPLC | Iyahambisana | |
Ukuncibilika | Incibilika ku-Dimethylsulfoxide, incibilika kancane ku-Ethanol ne-Acetonitrile, nge-pH encibilika emanzini | Iyahambisana |
Okuqukethwe kwamanzi(KF) | ≤ 1.00% | 0.42% |
Izinsalela ekushiseni | ≤ 0.10% | 0.05% |
Hi-eavyMethi | ≤ 20ppm | Iyahambisana |
I-Mesylate | 15.20%~18.20% | 15.90% |
Izincibilikisi Ezisele | I-Acetonitrile: ≤410ppm | ND |
I-acetone: ≤5000ppm | ND | |
I-Tetrahydrofuran: ≤720ppm | ND | |
RejabuleSizinto | Ubuningi bokungcola okukodwa: ≤0.20% | 0.17% |
Ukungcola okuphelele: ≤1.00% | 0.25% | |
Usayizi Wezinhlayiyana | I-D90: ≤100μm | 57.97% |
Asho (isisekelo se-HPLC ekomisweni) | 98.00%~102.00% | 99.80% |
Izinga Lereferensi | In-house Standard |